Awọn oògùn Antithyroid ti a lo lati ṣe itọju Arun Graves ati Hyperthyroidism
Awọn oloro Antithyroid - tun tọka si bi thioamides - awọn oogun ti o ṣe abojuto tairodura ti o nira (hyperthyroidism) nipasẹ didi iṣan tairodu gland lati ṣe awọn homonu tairodu. Ni itọju ti tairodu ti overactive, eyi ti o jẹ julọ julọ lati inu ipo autoimmune ti a mọ ni arun Graves, o jẹ pataki lati fa fifalẹ iṣan ti iṣan ti awọn homonu tairodu, paapaa awọn thymonia (T4) ti homonu ati triiodothyronine (T3).
Awọn iṣẹ oloro Antithyroid ṣiṣẹ nipasẹ ṣiṣe ti o nira sii fun ara lati lo iodine, nitorinaa ṣe idaduro ifarahan awọn homonu tairodu ninu ẹṣẹ.
Antityroid oògùn ailera jẹ ọkan ninu awọn itọju fun hyperthyroidism ati aisan Graves. Awọn itọju miiran pẹlu ipilẹ iyọ ti o ni iidine (RAI) ti ipanilara ati igbesẹ ti isẹ-ara tabi apakan ti ẹjẹ tairodu .
Awọn oloro meji antithyroid ti o wa ni Orilẹ Amẹrika wa: propylthiouracil (PTU) ati methimazole. Ni Amẹrika, a n pe methimazole ni oògùn antithyroid to fẹ julọ ni ọpọlọpọ awọn ipo.
Methimazole, ti a npe ni thiamazole, a ma mu ki tairodu kuro lati lilo iodine lati mu homonu tairodu. O gba gbogbo igba bi iwọn lilo lẹẹkan fun ọjọ kan.
Ti lo oògùn ni gbogbo agbaye. Ni Orilẹ Amẹrika, Tapazole jẹ orukọ orukọ nikan ti antithyroid oògùn methimazole. Awọn nọmba ti awọn onisọpọ jeneriki ti methimazole wa.
Tapazole
Tapazole jẹ orukọ iyasọtọ ti methimazole , oògùn antithyroid ti Ọba Pharmaceuticals ti ṣe, Inc. Ti Tapazole Fọwọsi ni FDA ni ọdun 2000.
Tapazole Eroja : methimazole USP; lactose monohydrate; iṣuu magnẹsia stearate; sitashi (oka); aṣoju ti o ni idaniloju; ati talc.
Awọn Agbara Wa : 5 miligiramu ati 10 miligiramu
Generic Methimazole (nipasẹ Sandoz)
Sandoz, ẹgbẹ kan ti Orilẹ-ede Awọn Ile-iṣẹ Novartis, n ṣe akọọlẹ methimazole kan. O ti fọwọsi nipasẹ FDA ni ọdun 2001.
Sandoz Methimazole Eroja: methimazole USP; lactose monohydrate; iṣuu magnẹsia stearate; sitashi (oka); ati talc.
Awọn Agbara Wa: 5 miligiramu ati 10 miligiramu
Generic Methimazole (nipasẹ Cedar Pharmaceuticals LLC)
Cedar Pharmaceuticals LLC fun awọn olupese kan jakejado methimazole ti a pin nipasẹ Awọn Iwadi Iwadi United Research. Ipadasilẹ FDA ti gba ni ọdun 2005.
Cedar Pharmaceuticals Methimazole Eroja: methimazole USP; ṣe idaraya monohydrate; iṣuu magnẹsia stearate; ọdunkun ilẹkun; ati talc.
Agbara Wa: 5 miligiramu, 10 miligiramu, 15 miligiramu, 20 miligiramu
Generic Methimazole (nipasẹ Activis Totowa)
Awọn oluṣeto Totowa LLC Awọn oluṣelọpọ generic methimazole ati ifọwọsi FDA ni a gba ni ọdun 2007.
Iṣẹ Methimazole Eroja methimazole USP; lactose monohydrate; iṣuu magnẹsia stearate; sitashi pregelatinized; ati talc.
Awọn agbara wa: 5 miligiramu ati 10 miligiramu
Generic Methimazole (nipasẹ Awọn Ile-ẹkọ Imudanilogbo Caraco)
Carabo Pharmaceutical Laboratories, Ltd. n ṣe akọọlẹ methimazole ti a fọwọsi nipasẹ FDA ni ọdun 2007.
Caraco Methimazole Eroja: methimazole USP; lactose monohydrate; povidone; talc; croscarmellose; iṣuu magnẹsia stearate; ati sitashi.
Awọn Agbara Wa: 5mg ati 10mg
Generic Methimazole (nipasẹ Awọn Ile-iṣẹ Imudaniloju)
Nipa Awọn ile-iwosan Awọn iṣelọpọ n ṣe akọọlẹ methimazole kan.
Eroja: methimazole USP; lactose monohydrate; iṣuu magnẹsia stearate; ọkà ọka; ati talc.
Awọn Agbara Wa: 5 miligiramu ati 10 miligiramu
Awọn orisun:
Daily Med, US Food and Drug Administration Medication Database.
Awọn ibaraẹnisọrọ abojuto FDA Drug: Iboju Titun Titun lori Ipa Ẹtan Tii Pẹlu Propylthiouracil, Kẹrin 21, 2010
Ross, Douglas MD, "Alaye alaisan: Awọn antithyroid oloro," UpToDate . Imudojuiwọn ti o kẹhin: Kọkànlá Oṣù 13, 2009
Iroyin afikun nipa: Leslie Blumenberg